Примери за използване на Metabolisers на Английски и техните преводи на Български
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Poor metabolisers(PM).
CYP2D6 extensive/poor metabolisers.
In poor metabolisers(PMs).
Some of the children were found to be CYP2D6 ultra-rapid metabolisers.
CYP2D6 poor metabolisers.
Хората също превеждат
Poor metabolisers of CYP2D6.
In patients for whom it is known they are CYP2D6 ultra-rapid metabolisers”.
Intermediate metabolisers(IM).
Extensive CYP 2D6 metabolisers convert risperidone rapidly into 9-hydroxy-risperidone, whereas poor CYP 2D6 metabolisers convert it much more slowly.
Ultra-rapid metabolisers(UM).
Extensive CYP 2D6 metabolisers convert risperidone rapidly into 9-hydroxy-risperidone, whereas poor CYP 2D6 metabolisers convert it much more slowly.
O Caution should be used with moderate CYP2D6 inhibitors in intermediate metabolisers(IMs) and extensive metabolisers(EMs).
Extensive metabolisers CYP2C9*1*1.
The recommended dose is 84 mg eliglustat twice daily in CYP2D6 intermediate metabolisers(IMs) and extensive metabolisers(EMs).
Known poor metabolisers of CYP2D6 or CYP2C19.
Individuals are normally classified as poor(PM), extensive(EM)or ultrarapid metabolisers(UM), depending on the activity of the enzyme.
O In CYP2D6 intermediate metabolisers(IMs) or poor metabolisers(PMs) with any degree of hepatic impairment, Cerdelga is not recommended.
Caution should be used with strong ormoderate CYP3A inhibitors in intermediate metabolisers(IMs) and extensive metabolisers(EMs).
In CYP2D6 intermediate metabolisers(IMs) or poor metabolisers(PMs) with any degree of hepatic impairment, eliglustat is not recommended(see sections 4.4 and 5.2).
This included contraindication in patients of any age known to be CYP2D6 ultra-rapid metabolisers and in women of all ages who are breastfeeding.
No substantial differences in active metabolite exposure and mean inhibition of platelet aggregation(IPA) were observed between ultrarapid,extensive and intermediate metabolisers.
Intermediate metabolisers CYP2C9*2*2.
Clinical experience in CYP2D6 poor metabolisers(PMs) and ultra-rapid metabolisers(URMs).
Cerdelga is indicated in patients who are CYP2D6 poor metabolisers(PMs), intermediate metabolisers(IMs) or extensive metabolisers(EMs).
O Eliglustat is contraindicated in patients who are CYP2D6 intermediate metabolisers(IMs) or extensive metabolisers(EMs) who are taking a strong or moderate CYP2D6 inhibitor concomitantly with a strong or moderate CYP3A inhibitor.