What is the translation of " PARTIAL AGONIST " in Serbian?

• parcijalni agonist

Examples of using Partial agonist in English and their translations into Serbian

Anandamide, similar to THC, is a partial agonist of CB1R.
Анандамид, сличан ТХЦ-у, делимични је агонист ЦБ1Р.

It is a partial agonist of the A4B2 nicotinic acetylcholine receptor.
То је парцијални агонист алфа-4 бета-2( α4β2) никотинског ацетилхолинског рецептора.

It also functions as a 5-HT1A receptor weak partial agonist/ antagonist.
On takođe funkcioniše kao slab parcijalni agonist/ antagonist 5-HT1A receptora.

It is a partial agonist selective for alpha-4, beta-2 nicotinic acetylcholine receptor subtypes.
То је парцијални агонист алфа-4 бета-2( α4β2) никотинског ацетилхолинског рецептора.

DCI has low potency and acts as a partial agonist/antagonist at these receptors.
DCI ima nisku potentnost i deluje kao parcijalni agonist/ antagonist na tim receptorima.

It has a unique pharmacology: it is a selective β1 receptor antagonist, but a β2 receptor partial agonist.
On ima jedinstvenu farmakologiju: on je selektivan antagonist β1 receptora, i parcijalni agonist β2 receptora.

ACC is also an exogenous partial agonist of the mammalian NMDA receptor.
ACC takođe nefiziološki parcijalni agonist NMDA receptora sisara.

Fenoldopam mesylate(Corlopam) is a drug and synthetic benzazepine derivative which acts as a selective D1 receptor partial agonist.
Fenoldopam( Korlopam) je lek i sintetički derivat benzazepina koji deluje kao periferni selektivni parcijalni agonist/ antagonist D1 receptora.

Additionally, it is a partial agonist of 5-HT1A receptors.
On takođe funkcioniše kao slab parcijalni agonist/ antagonist 5-HT1A receptora.

It is a partial agonist at the cannabinoid receptor CB1, producing a maximal stimulation of 58.3% with a Ki of 8.45nM.
O-1238 je parcijalni agonist kanabinoidnog receptora CB1, sa maksimalnom stimulacijom od 58. 3% i Ki vrednošću od 8, 45 nM.

It has also been shown to function as a 5-HT1A receptor partial agonist and 5-HT2A and 5-HT2B receptor antagonist.
On takođe deluje kao parcijalni agonist 5-HT1A receptora i antagonist 5-HT2A i 5-HT2B receptora.

In the presence of progesterone, mifepristone acts as a competitive progesterone receptor antagonist(in the absence of progesterone, mifepristone acts as a partial agonist).
U prisustvu progesterona, mifepriston dejstvuje kao kompetitivni antagonist progesteronskog receptora( u odsustvu progesterona, mifepriston dejstvuje kao parcijalni agonist).

Cisapride and tegaserod are 5-HT4 receptor partial agonists that were used to treat disorders of gastrointestinal motility.
Cisaprid i Tegaserod su parcijalni agonisti 5-HT4 receptora koji se koriste za tretiranje poremećaja gastrointestinalne motilnosti.

Br-APB is a synthetic compound that acts as a selective D1 agonist, with the(R)-enantiomer being a potent full agonist, while the(S) enantiomer retains its D1 selectivity but is a weak partial agonist.
( R)- enantiomer je potentan pun agonist, dok( S) enantiomer ima D1 selektivnost, ali je slab parcijalni agonist.

Piclozotan(SUN-N4057) is a selective 5-HT1A receptor partial agonist, which has neuroprotective effects in animal studies.
Piklozotan( SUN-N4057) je selektivni parcijalni agonist 5-HT1A receptora, koji ima neuroprotektivno dejstvo u životinjskim studijama.

Partial agonists(such as buspirone, aripiprazole, buprenorphine, or norclozapine) also bind and activate a given receptor, but have only partial efficacy at the receptor relative to a full agonist, even at maximal receptor occupancy.
Parcijalni agonisti( kao što su buspiron, aripiprazol, buprenorfin, ili norklozapin) se takođe vezuju i aktiviraju dati receptor, ali oni imaju samo parcijalnu efikasnost u odnosu na pun agonist..

Rivanicline(TC-2403, RJR-2403,(E)-metanicotine) is a drug which acts as a partial agonist at neural nicotinic acetylcholine receptors.
Rivaniklin( TC-2403, RJR-2403,( E)- metanikotin) je lek koji deluje kao parcijalni agonist neuronskih nikotinskih acetilholinskih receptora.

Aripiprazole is believed to act mostly as a"partial agonist" of dopamine and 5-hydroxytryptamine neurotransmitter receptors(also called serotonin).
Верује се да арипипразол делује углавном као" делимични агонист" допаминских и 5-хидрокситриптаминских неуротрансмитерских рецептора( који се називају и серотонин).

They are ligands and include receptor agonists and receptor antagonists, as well as receptor partial agonists, inverse agonists, and allosteric modulators.
То су лиганди и укључују агонисте рецептора и антагонисте рецептора, као и парцијалне агонисте, инверзне агонисте и алостерне модулаторе рецептора.

Some of the atypical antipsychotics like lurasidone and aripiprazole are also partial agonists at the 5-HT1A receptor and are sometimes used in low doses as augmentations to standard antidepressants like the selective serotonin reuptake inhibitors(SSRIs).
Neki od atipičnih antipsihotika kao što je aripiprazol su takođe parcijalni agonisti 5-HT1A receptora i ponekad se koriste u niskim dozama kao zamena za standardne antidepresive kao što su selektivni inhibitori preuzimanja serotonina( SSRI).

It also has affinity for the 5-HT2A, 5-HT2B, and 5-HT2C receptors(EC50 values= 466 nM, 40 nM, and 2.3 nM, respectively), and acts as a full agonist at 5-HT2B and as a partial agonist at 5-HT2C, while its affinity for 5-HT2A is probably too low to be significant.
On takođe ima visok afinitet za 5-HT2A, 5-HT2B, i 5-HT2C receptore( EC50 vrednosti= 466 nM, 40 nM, i 2. 3 nM, respektivno), i deluje kao pun agonist na 5-HT2B i kao parcijalni agonist na 5-HT2C, dok je njegov afinitet za 5-HT2A verovatno suviše nizak da bi bio značajan.

Tandospirone acts as a potent and selective 5-HT1A receptor partial agonist, with a Ki affinity value of 27± 5 nM and approximately 55 to 85% intrinsic activity.
Tandospiron deluje kao potentan i selektivan parcijalni agonist 5-HT1A receptora, sa Ki afinitetom od 27 ± 5 nM i aproksimativno 55-85% intrinsične aktivnosti.

Role in memory and learning Activation of the 5-HT2A receptor is necessary for the effects of the"classic" psychedelics like LSD, psilocin and mescaline, which act as full or partial agonists at this receptor, and represent the three main classes of 5-HT2A agonists, the ergolines, tryptamines and phenethylamines, respectively.
Aktivacija 5-HT2A receptora je neophodna za dejstvo„ klasičnih“ psihodelika kao što su LSD, psilocin i meskalin, koji deluju kao puni ili parcijalni agonisti ovog receptora, i predstavljaju tri glavne klase 5-HT2A agonista, ergolina, triptamina i fenetilamina, respektivno.